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GPCR & Ion Channel Stable Cell Line Collection

GenScript offers a wide collection of GPCR and ion channel stable cell lines for compound screening/profiling services. In addition, you can purchase the stable cell lines and perform a screening project in-house. Furthermore, customized reagent preparation services are available upon your specifications: Ready-to-UseTM Frozen Cells, Membrane Preparations, and Custom Stable Cell Line Service.

GPCRs

Cat. No.
Cell Line
GPCR Family
Receptor
Price (USD)
Selected
CHO-K1/M1 Acetylcholine (muscarinic) M1 / CHRM1
$11600.00
CHO-K1/M2/Gα15 Acetylcholine (muscarinic) M2 / CHRM2
$11600.00
CHO-K1/M3 Acetylcholine (muscarinic) M3 / CHRM3
$11600.00
CHO-K1/M4/Gα15 Acetylcholine (muscarinic) M4 / CHRM4
$11600.00
CHO-K1/M5 Acetylcholine (muscarinic) M5 / CHRM5
$11600.00
CHO-K1/ADORA1/Gα15 Adenosine ADORA1
$11600.00
CHO-K1/ADORA2A/Gα15 Adenosine ADORA2A
$11600.00
CHO-K1/ADORA2B/Gα15 Adenosine ADORA2B
$11600.00
CHO-K1/ADRA1A Adrenoceptors ADRA1A
$11600.00
CHO-K1/ADRA1B Adrenoceptors ADRA1B
$11600.00
CHO-K1/ADRA1D Adrenoceptors ADRA1D
$11600.00
CHO-K1/ADRA2A/Gα15 Adrenoceptors ADRA2A
$11600.00
CHO-K1/ADRA2C/Gα15 Adrenoceptors ADRA2C
$11600.00
CHO-K1/ADRB1/Gα15 Adrenoceptors ADRB1
$11600.00
CHO-K1/ADRB2/Gα15 Adrenoceptors ADRB2
$11600.00
293/ADRB3/CRE-Luc Adrenoceptors ADRB3
$11600.00
CHO-K1/C5a/Gα15 Anaphylotoxin C5a / C5AR1
$11600.00
293T/AT1 Angiotensin AT1
$11600.00
CHO-K1/AT2/Gqi5 Angiotensin AT2
$11600.00
CHO-K1/AGTRL1/Gα15 Apelin AGTRL1
$11600.00
CHO-K1/GPBAR1 Bile acid GPBAR1
$11600.00
CHO-K1/BB1 Bombesin BB1
$11600.00
CHO-K1/BB2 Bombesin BB2
$11600.00
CHO-K1/BB3 Bombesin BB3
$11600.00
CHO-K1/B2/Gα15 Bradykinin B2
$11600.00
CHO-K1/CNR1/Gα15 Cannabinoid CNR1 / CB1
$11600.00
CHO-K1/CNR2 Cannabinoid CNR2 / CB2
$11600.00
CHO-K1/CMKLR1/Gα15 Chemoattractant ChemR23 / CMKLR1
$11600.00
CHO-K1/CCKA/Gα15 Cholecystokinin CCKA
$11600.00
CHO-K1/CCKB Cholecystokinin CCKB
$11600.00
CHO-K1/D1 Dopamine D1 / DRD1
$11600.00
M00348
293/D1/CRE-Luc Dopamine D1 / DRD1
$11600.00
Coming soon
CHO-K1/D2/Gα15 Dopamine D2 / DRD2
$11600.00
CHO-K1/D2S/Gα15 Dopamine D2S / DRD2S
$11600.00
CHO-K1/D5/Gα15 Dopamine D5 / DRD5
$11600.00
CHO-K1/EDNRA Endothelin EDNRA
$11600.00
CHO-K1/EDNRB Endothelin EDNRB
$11600.00
CHO-K1/GPR120/Gα15 Free Fatty Acid GPR120
$11600.00
CHO-K1/FFA1/Gα15 Free Fatty Acid FFA1 / GPR40
$11600.00
CHO-K1/FFA2/Gα15 Free Fatty Acid FFA2 / GPR43
$11600.00
CHO-K1/GAL1/Gα15 Galanin GAL1
$11600.00
CHO-K1/GAL2 Galanin GAL2
$11600.00
CHO-K1/GHSR Ghrelin GHSR
$11600.00
CHO-K1/GNRHR/Gα15 Gonadotropin-releasing Hormone GNRHR
$11600.00
293/H1 Histamine H1
$11600.00
CHO-K1/H2/Gα15 Histamine H2
$11600.00
CHO-K1/H3/Gα15 Histamine H3
$11600.00
CHO-K1/H4/Gα15 Histamine H4
$11600.00
CHO-K1/KiSS1 KiSS1-derived Peptide KiSS1 / GPR54
$11600.00
CHO-K1/LTB4/Gα15 Leukotriene LTB4
$11600.00
CHO-K1/MRGPRX2 Mas-related gene MRGX2 / MRGPRX2
$11600.00
293/MCH1 Melanin-concentrating Hormone MCH1
$11600.00
CHO-K1/MCH2 Melanin-concentrating Hormone MCH2
$11600.00
CHO-K1/MC2/Gα15 Melanocortin MC2
$11600.00
CHO-K1/MC3/Gα15 Melanocortin MC3
$11600.00
293/MC3/CRE-Luc Melanocortin MC3
$11600.00
CHO-K1/MC4/Gα15 Melanocortin MC4
$11600.00
CHO-K1/MC5/Gα15 Melanocortin MC5
$11600.00
CHO-K1/MT1/Gα15 Melatonin MT1
$11600.00
CHO-K1/MT2/Gα15 Melatonin MT2
$11600.00
CHO-K1/MTLR/Gα15 Motilin MTLR
$11600.00
CHO-K1/NMU1 Neuromedin U NMU1
$11600.00
293T/NMU2 Neuromedin U NMU2
$11600.00
CHO-K1/NPFF1/Gα15 Neuropeptide FF NPFF1 / GPR147
$11600.00
CHO-K1/NPS1a/Gα15 Neuropeptide S NPS1a
$11600.00
CHO-K1/NPS1b/Gα15 Neuropeptide S NPS1b
$11600.00
M00192
CHO-K1/NPY1/Gα15 Neuropeptide Y NPY1
$11600.00
Coming soon
M00430
293/NPY1 Neuropeptide Y NPY1
$11600.00
Coming soon
M00237
CHO-K1/NPY4/Gα15 Neuropeptide Y NPY4 / PPYR1
$11600.00
Coming soon
CHO-K1/NTS1 Neurotensin NTS1
$11600.00
CHO-K1/NIACR1/Gα15 Nicotinic Acid NIACR1 / GPR109A
$11600.00
CHO-K1/FPR1/Gα15 N-Formyl Peptide FPR1
$11600.00
CHO-K1/FPRL1/Gα15 N-Formyl Peptide FPRL1
$11600.00
CHO-K1/OPRD1/Gα15 Opioid OPRD1
$11600.00
CHO-K1/OPRK1/Gα15 Opioid OPRK1
$11600.00
CHO-K1/OPRL1/Gα15 Opioid OPRL1
$11600.00
CHO-K1/OPRM1/Gα15 Opioid OPRM1
$11600.00
CHO-K1/OX1 Orexin OX1
$11600.00
CHO-K1/OX2 Orexin OX2
$11600.00
CHO-K1/OXTR Oxytocin OT / OXTR
$11600.00
CHO-K1/GPR103/Gα15 Peptide P518 GPR103
$11600.00
CHO-K1/PTAFR Platelet Activating Factor PAF / PTAFR
$11600.00
CHO-K1/PRLHR Prolactin Releasing Peptide PRLHR
$11600.00
CHO-K1/DP2/Gα15 Prostanoid DP2 / GPR44
$11600.00
293/FP/Gα15 Prostanoid FP / PTGFR
$11600.00
293/PTGER1 Prostanoid EP1 / PTGER1
$11600.00
CHO-K1/PTGER2/Gα15 Prostanoid EP2 / PTGER2
$11600.00
CHO-K1/IP1/Gα15 Prostanoid IP1 / PTGIR
$11600.00
293/TP Prostanoid TP / TBXA2R
$11600.00
CHO-K1/PAR2/Gα15 Proteinase-activated Receptor PAR2 / F2RL1
$11600.00
CHO-K1/PAR4 Proteinase-activated Receptor PAR4 / F2RL3
$11600.00
CHO-K1/GPR68/Gα15 Proton-sensor GPR68
$11600.00
M00250
1321N1/P2Y1 Purinergic P2Y1
$11600.00
Coming soon
1321N1/P2Y2 Purinergic P2Y2
$11600.00
1321N1/P2Y4 Purinergic P2Y4
$11600.00
1321N1/P2Y6 Purinergic P2Y6
$11600.00
1321N1/P2Y11 Purinergic P2Y11
$11600.00
1321N1/P2Y12 Purinergic P2Y12
$11600.00
CHO-K1/5-HT1A/Gα15 Serotonin 5-HT1A / HTR1A
$11600.00
CHO-K1/5-HT2A Serotonin 5-HT2A / HTR2A
$11600.00
CHO-K1/5-HT2B Serotonin 5-HT2B / HTR2B
$11600.00
CHO-K1/5-HT2C Serotonin 5-HT2C / HTR2C
$11600.00
HEK293/5-HT2C Serotonin 5-HT2C / HTR2C
$11600.00
CHO-K1/5-HT4/Gqi5 Serotonin 5-HT4 / HTR4
$11600.00
M00423
293/5-HT7/CRE-Luc Serotonin 5-HT7 / HTR7
$11600.00
Coming soon
CHO-K1/SST2/Gα15 Somatostatin SST2
$11600.00
CHO-K1/SST3/Gα15 Somatostatin SST3
$11600.00
CHO-K1/SST4/Gα15 Somatostatin SST4
$11600.00
CHO-K1/SST5/Gα15 Somatostatin SST5
$11600.00
CHO-K1/NK1 Tachykinin NK1 / TACR1
$11600.00
CHO-K1/NK2 Tachykinin NK2 / TACR2
$11600.00
CHO-K1/NK3 Tachykinin NK3 / TACR3
$11600.00
CHO-K1/TRH1 Thyrtropin-releasing Hormone TRH1
$11600.00
CHO-K1/UT2/Gα15 Urotensin UT2
$11600.00
CHO-K1/V1A Vasopressin V1A / AVPR1A
$11600.00
CHO-K1/V1B Vasopressin V1B / AVPR1B
$11600.00
CHO-K1/V2/Gα15 Vasopressin V2 / AVPR2
$11600.00
M00350
CHO-K1/AMY1/CRE-Luc Calcitonin AMY1 (RAMP1+CT)
$11600.00
Coming soon
CHO-K1/CT/Gα15 Calcitonin CALCR / CT
$11600.00
CHO-K1/CRF1/Gα15 Corticotropin Releasing Factor CRF1
$11600.00
CHO-K1/CRF2/Gα15 Corticotropin Releasing Factor CRF2
$11600.00
CHO-K1/GCGR/Gα15 Glucagon GCGR
$11600.00
293/GHRH/Gα15 Glucagon GHRH
$11600.00
CHO-K1/GLP2/Gα15 Glucagon GLP2
$11600.00
CHO-K1/SCTR/Gα15 Glucagon SCTR
$11600.00
CHO-K1/PTH1/Gα15 Parathyroid Hormone PTH1
$11600.00
293/PTH2/CRE-Luc Parathyroid Hormone PTH2
$11600.00
CHO-K1/PAC1/Gα15 VIP / PACAP PAC1
$11600.00
CHO-K1/VPAC1/Gα15 VIP / PACAP VPAC1
$11600.00
CHO-K1/VPAC2/Gα15 VIP / PACAP VPAC2
$11600.00
CHO-K1/CASR Calcium-sensor CASR
$11600.00
CHO-K1/GRM2/Gα15 Glutamate mGlu2 / GRM2
$11600.00
CHO-K1/CRE-Luc Control  
$11600.00
293/CRE-Luc Control  
$11600.00
M00257
CHO-K1/Gα15 Control  
$11600.00
Coming soon
CHO-K1/Gqi5 Control  
$11600.00

All the GPCRs are available as Ready-to-UseTM frozen cells.
A part of the GPCRs are available as Membrane Preparations.

Ion Channels

Name
Type
Channel
Accession Number
CHO-K1/hERG Potassium, voltage-gated hERG (Kv11.1)
NM_000238.2
HEK293/hERG Potassium, voltage-gated hERG (Kv11.1)
NM_000238.2
HEK293/hKv1.5 Potassium, voltage-gated hKv1.5
NM_002234
HEK293/hKv4.2 Potassium, voltage-gated hKv4.2
NM_012281
HEK293/hNav1.5 Sodium, voltage-gated hNav1.5
NM_000335
HEK293/hNav1.7 Sodium, voltage-gated hNav1.7
NM_002977

Custom Stable Cell Line Services:

Cat. No. Service
Price (USD)
SC1394
Custom Stable Cell Line Service

Related Services:


Email: bioassay@genscript.com
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