Class | Ligand Type | GPCR Family | Receptor | Cell Line | Cat. No. |
A | Non-peptide | Acetylcholine (muscarinic) | M1 / CHRM1 | CHO-K1/M1 | |
A | Non-peptide | Acetylcholine (muscarinic) | M2 / CHRM2 | CHO-K1/M2/Gα15 | |
A | Non-peptide | Acetylcholine (muscarinic) | M3 / CHRM3 | CHO-K1/M3 | |
A | Non-peptide | Acetylcholine (muscarinic) | M4 / CHRM4 | CHO-K1/M4/Gα15 | |
A | Non-peptide | Acetylcholine (muscarinic) | M5 / CHRM5 | CHO-K1/M5 | |
A | Non-peptide | Adenosine | ADORA1 | CHO-K1/ADORA1/Gα15 | |
A | Non-peptide | Adenosine | ADORA1 | 293/ADORA1/Gα15 | |
A | Non-peptide | Adenosine | ADORA2A | CHO-K1/ADORA2A/Gα15 | |
A | Non-peptide | Adenosine | ADORA2B | CHO-K1/ADORA2B/Gα15 | |
A | Non-peptide | Adenosine | ADORA3 | CHO-K1/ADORA3/Gqi5 | |
A | Non-peptide | Adrenoceptors | ADRA1A | CHO-K1/ADRA1A | |
A | Non-peptide | Adrenoceptors | ADRA1B | CHO-K1/ADRA1B | |
A | Non-peptide | Adrenoceptors | ADRA1D | CHO-K1/ADRA1D | |
A | Non-peptide | Adrenoceptors | ADRA2A | CHO-K1/ADRA2A/Gα15 | |
A | Non-peptide | Adrenoceptors | ADRA2B | CHO-K1/ADRA2B/Gqi5 | |
A | Non-peptide | Adrenoceptors | ADRA2C | CHO-K1/ADRA2C/Gα15 | |
A | Non-peptide | Adrenoceptors | ADRB1 | CHO-K1/ADRB1/Gα15 | |
A | Non-peptide | Adrenoceptors | ADRB2 | CHO-K1/ADRB2/Gα15 | |
A | Non-peptide | Adrenoceptors | ADRB3 | 293/ADRB3/CRE-Luc | |
A | Peptide | Anaphylotoxin | C5a / C5AR1 | CHO-K1/C5a/Gα15 | |
A | Peptide | Angiotensin | AT1 | 293T/AT1 | |
A | Peptide | Angiotensin | AT1 | HEK293/AT1 | |
A | Peptide | Apelin | AGTRL1 | CHO-K1/AGTRL1/Gα15 | |
A | Non-peptide | Bile acid | GPBAR1 | CHO-K1/GPBAR1 | |
A | Peptide | Bombesin | BB1 / NMBR | CHO-K1/BB1 | |
A | Peptide | Bombesin | BB2 / GRPR | CHO-K1/BB2 | |
A | Peptide | Bombesin | BB3 / BRS3 | CHO-K1/BB3 | |
A | Peptide | Bradykinin | B1 / BDKRB1 | CHO-K1/B1/Gα15 | M00482 |
A | Peptide | Bradykinin | B2 / BDKRB2 | CHO-K1/B2/Gα15 | |
A | Non-peptide | Cannabinoid | CB1 / CNR1 | CHO-K1/CB1/Gα15 | |
A | Non-peptide | Cannabinoid | CB2 / CNR2 | CHO-K1/CB2 | |
A | Peptide | Chemoattractant | ChemR23 / CMKLR1 | CHO-K1/CMKLR1/Gα15 | |
A | Peptide | Cholecystokinin | CCKA | CHO-K1/CCKA/Gα15 | |
A | Peptide | Cholecystokinin | CCKB | CHO-K1/CCKB | |
A | Non-peptide | Dopamine | D1 / DRD1 | CHO-K1/D1 | |
A | Non-peptide | Dopamine | D2 / DRD2 | CHO-K1/D2/Gα15 | |
A | Non-peptide | Dopamine | D2S / DRD2S | CHO-K1/D2S/Gα15 | |
A | Non-peptide | Dopamine | D4 / DRD4 | 293/D4 | M00477 |
A | Non-peptide | Dopamine | D5 / DRD5 | CHO-K1/D5/Gα15 | |
A | Peptide | Endothelin | EDNRA | CHO-K1/EDNRA | |
A | Peptide | Endothelin | EDNRB | CHO-K1/EDNRB | |
A | Non-peptide | Free Fatty Acid | FFA1 / GPR40 | CHO-K1/FFA1/Gα15 | |
A | Non-peptide | Free Fatty Acid | FFA2 / GPR43 | CHO-K1/FFA2/Gα15 | |
A | Peptide | Galanin | GAL1 | CHO-K1/GAL1/Gα15 | |
A | Peptide | Galanin | GAL2 | CHO-K1/GAL2 | |
A | Peptide | Ghrelin | GHSR | CHO-K1/GHSR | |
A | Peptide | Gonadotropin-releasing Hormone | GNRHR | CHO-K1/GNRHR/Gα15 | |
A | Non-peptide | Histamine | H1 | 293/H1 | |
A | Non-peptide | Histamine | H2 | CHO-K1/H2/Gα15 | |
A | Non-peptide | Histamine | H3 | CHO-K1/H3/Gα15 | |
A | Non-peptide | Histamine | H4 | CHO-K1/H4/Gα15 | |
A | Peptide | KiSS1-derived Peptide | KiSS1 / GPR54 | CHO-K1/KiSS1 | |
A | Non-peptide | Leukotriene | CysLT1 | CHO-K1/CysLT1/Gα15 | |
A | Non-peptide | Leukotriene | CysLT2 | CHO-K1/CysLT2 | |
A | Non-peptide | Leukotriene | LTB4 | CHO-K1/LTB4/Gα15 | |
A | Non-peptide | Leukotriene | OXE / OXER1 | CHO-K1/OXE-Flag/Gα15 | M00488 |
A | Non-peptide | Lysophospholipid | EDG4 / LPA2 | RH7777/EDG4 | |
A | Non-peptide | Lysophospholipid | EDG6 / S1P4 | RH7777/EDG6 | M00465 |
A | Peptide | Melanin-concentrating Hormone | MCH1 | 293/MCH1 | |
A | Peptide | Melanin-concentrating Hormone | MCH2 | CHO-K1/MCH2 | |
A | Peptide | Melanocortin | MC2 | CHO-K1/MC2/Gα15 | |
A | Peptide | Melanocortin | MC3 | CHO-K1/MC3/Gα15 | |
A | Peptide | Melanocortin | MC3 | 293/MC3/CRE-Luc | |
A | Peptide | Melanocortin | MC4 | CHO-K1/MC4/Gα15 | |
A | Peptide | Melanocortin | MC5 | CHO-K1/MC5/Gα15 | |
A | Peptide | Melatonin | MT1 / MTNR1A | CHO-K1/MT1/Gα15 | |
A | Peptide | Melatonin | MT2 / MTNR1B | CHO-K1/MT2/Gα15 | |
A | Peptide | Motilin | MTLR | CHO-K1/MTLR/Gα15 | |
A | Peptide | Neuromedin U | NMU1 | CHO-K1/NMU1 | |
A | Peptide | Neuromedin U | NMU2 | 293T/NMU2 | |
A | Peptide | Neuropeptide B/W | NPBW1 / GPR7 | CHO-K1/NPBW1/Gα15 | |
A | Peptide | Neuropeptide FF | NPFF1 / GPR147 | CHO-K1/NPFF1/Gα15 | |
A | Peptide | Neuropeptide FF | NPFF2 / GPR74 | CHO-K1/NPFF2/Gα15 | |
A | Peptide | Neuropeptide S | NPS1a | CHO-K1/NPS1a/Gα15 | |
A | Peptide | Neuropeptide S | NPS1b | CHO-K1/NPS1b/Gα15 | |
A | Peptide | Neuropeptide Y | NPY1 | CHO-K1/NPY1/Gα15 | M00192 |
A | Peptide | Neuropeptide Y | NPY1 | 293/NPY1 | M00430 |
A | Peptide | Neuropeptide Y | NPY2 | CHO-K1/NPY2/Gqi5 | |
A | Peptide | Neuropeptide Y | NPY4 / PPYR1 | CHO-K1/NPY4/Gα15 | |
A | Peptide | Neurotensin | NTS1 | CHO-K1/NTS1 | |
A | Non-peptide | Nicotinic Acid | NIACR1 / GPR109A | CHO-K1/NIACR1/Gα15 | |
A | Peptide | N-Formyl Peptide | FPR1 | CHO-K1/FPR1/Gα15 | |
A | Peptide | N-Formyl Peptide | FPRL1 | CHO-K1/FPRL1/Gα15 | |
A | Peptide | Opioid | OPRD1 | CHO-K1/OPRD1/Gα15 | |
A | Peptide | Opioid | OPRK1 | CHO-K1/OPRK1/Gα15 | |
A | Peptide | Opioid | OPRL1 | CHO-K1/OPRL1/Gα15 | |
A | Peptide | Opioid | OPRM1 | CHO-K1/OPRM1/Gα15 | |
A | Peptide | Orexin | OX1 | CHO-K1/OX1 | |
A | Peptide | Orexin | OX2 | CHO-K1/OX2 | |
A | Peptide | Oxytocin | OT / OXTR | CHO-K1/OXTR | |
A | Peptide | Peptide P518 | GPR103 | CHO-K1/GPR103/Gα15 | |
A | Non-peptide | Platelet Activating Factor | PAF / PTAFR | CHO-K1/PTAFR | |
A | Peptide | Prolactin Releasing Peptide | PRLHR | CHO-K1/PRLHR | |
A | Non-peptide | Prostanoid | DP1 / PTGDR | CHO-K1/DP1/Gα15 | |
A | Non-peptide | Prostanoid | DP2 / GPR44 | CHO-K1/DP2/Gα15 | |
A | Non-peptide | Prostanoid | FP / PTGFR | 293/FP/Gα15 | |
A | Non-peptide | Prostanoid | EP1 / PTGER1 | 293/EP1 | |
A | Non-peptide | Prostanoid | EP2 / PTGER2 | CHO-K1/EP2/Gα15 | |
A | Non-peptide | Prostanoid | EP4 / PTGER4 | 293/EP4 | M00485 |
A | Non-peptide | Prostanoid | IP1 / PTGIR | CHO-K1/IP1/Gα15 | |
A | Non-peptide | Prostanoid | TP / TBXA2R | 293/TP | |
A | Peptide | Proteinase-activated Receptor | PAR2 / F2RL1 | CHO-K1/PAR2/Gα15 | |
A | Peptide | Proteinase-activa
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