GPCR & Ion Channel Stable Cell Line Collection
GenScript offers a wide selection of GPCR and ion channel stable cell lines exclusively for assay services. In addition, GenScript offers one-stop assay reagent preparations for your compound screening/profiling: Ready-to-UseTM Frozen Cells, Membrane Preparations, and Custom Stable Cell Line Service.
GPCRs
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| CHO-K1/M1 |
Acetylcholine (muscarinic) |
M1 / CHRM1 |
NM_000738 |
| CHO-K1/M3 |
Acetylcholine (muscarinic) |
M3 / CHRM3 |
NM_000740 |
| CHO-K1/M5 |
Acetylcholine (muscarinic) |
M5 / CHRM5 |
NM_012125 |
| CHO-K1/ADORA1/Gα15 |
Adenosine |
ADORA1 |
NM_000674 |
| CHO-K1/ADORA2B/Gα15 |
Adenosine |
ADORA2B |
NM_000675 |
| CHO-K1/ADRA1A |
Adrenoceptors |
ADRA1A |
NM_000680 |
| CHO-K1/ADRA1B |
Adrenoceptors |
ADRA1B |
NM_000679 |
| CHO-K1/ADRA1D |
Adrenoceptors |
ADRA1D |
NM_000678 |
| CHO-K1/ADRA2A/Gα15 |
Adrenoceptors |
ADRA2A |
NM_000681 |
| CHO-K1/ADRB1/Gα15 |
Adrenoceptors |
ADRB1 |
NM_000684 |
| CHO-K1/ADRB2/Gα15 |
Adrenoceptors |
ADRB2 |
NM_000024 |
| 293/ADRB3/CRE-Luc |
Adrenoceptors |
ADRB3 |
NM_000025 |
| CHO-K1/C5a/Gα15 |
Anaphylotoxin |
C5a / C5AR1 |
NM_001736 |
| CHO-K1/BB2 |
Bombesin |
BB2 |
NM_005314 |
| CHO-K1/BB3 |
Bombesin |
BB3 |
NM_001727 |
| CHO-K1/B2/Gα15 |
Bradykinin |
B2 |
NM_000623 |
| CHO-K1/CALCR/Gα15 |
Calcitonin |
CALCR |
NM_001742.2 |
| CHO-K1/CNR1/Gα15 |
Cannabinoid |
CNR1 / CB1 |
NM_016083 |
| CHO-K1/CMKLR1/Gα15 |
Chemoattractant |
CMKLR1 |
NM_004072 |
| CHO-K1/CCKA/Gα15 |
Cholecystokinin |
CCKA |
NM_000730 |
| CHO-K1/CCKB |
Cholecystokinin |
CCKB |
NM_176875 |
| CHO-K1/CRF1/Gα15 |
Corticotropin Releasing Factor |
CRF1 |
NM_004382 |
| CHO-K1/CRF2/Gα15 |
Corticotropin Releasing Factor |
CRF2 |
NM_001883 |
| CHO-K1/D2/Gα15 |
Dopamine |
D2 |
NM_000795 |
| CHO-K1/D2s/Gα15 |
Dopamine |
D2S |
NM_016574 |
| CHO-K1/D5/Gα15 |
Dopamine |
D5 |
NM_000798 |
| CHO-K1/EDNRA |
Endothelin |
EDNRA |
NM_000795 |
| CHO-K1/EDNRB |
Endothelin |
EDNRB |
NM_000115 |
| CHO-K1/GPR40-GFP |
Free Fatty Acid |
FFA1 / GPR40 |
NM_005303 |
| CHO-K1/GPR40/Gα15 |
Free Fatty Acid |
FFA1 / GPR40 |
NM_005303 |
| CHO-K1/GAL1/Gα15 |
Galanin |
GAL1 |
NM_001480 |
| CHO-K1/GAL2 |
Galanin |
GAL2 |
NM_003857 |
| CHO-K1/GHSR |
Ghrelin |
GHSR |
NM_198407 |
| 293/GHRH/Gα15 |
Glucagon |
GHRH |
NM_000823 |
| CHO-K1/GLP2/Gα15 |
Glucagon |
GLP2 |
NM_004246 |
| CHO-K1/SCTR/Gα15 |
Glucagon |
SCTR |
NM_002980 |
| 293/H1 |
Histamine |
H1 |
NM_000861 |
| CHO-K1/H2/Gα15 |
Histamine |
H2 |
NM_022304 |
| CHO-K1/H3/Gα15 |
Histamine |
H3 |
NM_007232 |
| CHO-K1/H4/Gα15 |
Histamine |
H4 |
NM_021624 |
| CHO-K1/KISS1 |
KiSS1-derived peptide |
KiSS1 / GPR54 |
NM_032551 |
| 293/MCH1 |
Melanin-concentrating Hormone |
MCH1 |
NM_005297 |
| CHO-K1/MCH2 |
Melanin-concentrating Hormone |
MCH2 |
NM_032503 |
| CHO-K1/MC2/Gα15 |
Melanocortin |
MC2 |
NM_000529 |
| CHO-K1/MC3/Gα15 |
Melanocortin |
MC3 |
NM_019888 |
| 293/MC3/CRE-Luc |
Melanocortin |
MC3 |
NM_019888 |
| CHO-K1/MC4/Gα15 |
Melanocortin |
MC4 |
NM_005912 |
| CHO-K1/MT2/Gα15 |
Melatonin |
MT2 |
NM_005959 |
| CHO-K1/NMU1 |
Neuromedin U |
NMU1 |
NM_006056 |
| CHO-K1/GPR103/Gα15 |
Neuropeptide |
GPR103 |
NM_198179 |
| CHO-K1/NPS1a/Gα15 |
Neuropeptide S |
NPS1a |
NM_207172 |
| CHO-K1/NTS1 |
Neurotensin |
NTS1 |
NM_002531 |
| CHO-K1/FPRL1/Gα15 |
N-Formyl Peptide |
FPRL1 |
NM_001462 |
| CHO-K1/OPRD1/Gα15 |
Opioid |
OPRD1 |
NM_000911 |
| CHO-K1/OPRK1/Gα15 |
Opioid |
OPRK1 |
NM_000912 |
| CHO-K1/OPRM1/Gα15 |
Opioid |
OPRM1 |
NM_000914 |
| CHO-K1/OX1 |
Orexin |
OX1 |
NM_001525 |
| CHO-K1/OX2 |
Orexin |
OX2 |
NM_001526 |
| CHO-K1/OXTR |
Oxytocin |
OT / OXTR |
NM_000916 |
| CHO-K1/PTH1/Gα15 |
Parathyroid Hormone |
PTH1 |
NM_000316 |
| 293/PTH2/CRE-Luc |
Parathyroid Hormone |
PTH2 |
NM_005048 |
| CHO-K1/PTAFR |
Platelet Activating Factor |
PAF / PTAFR |
NM_000952 |
| 293/FP/Gα15 |
Prostanoid |
FP / PTGFR |
NM_000952 |
| 293/PTGER1 |
Prostanoid |
EP1 / PTGER1 |
NM_000955.2 |
| CHO-K1/PTGER2/Gα15 |
Prostanoid |
EP2 / PTGER2 |
NM_000956 |
| CHO-K1/IP1/Gα15 |
Prostanoid |
IP1 / PTGIR |
NM_000960 |
| 293/TP |
Prostanoid |
TP / TBXA2R |
NM_001060 |
| CHO-K1/PAR4 |
Proteinase-activated Receptor |
PAR4 / F2RL3 |
NM_003950 |
| CHO-K1/5-HT1A/Gα15 |
Serotonin |
5-HT1A / HTR1A |
NM_000524 |
| CHO-K1/5-HT1D/Gα15 |
Serotonin |
5-HT1D / HTR1D |
NM_000864 |
| CHO-K1/5-HT2A |
Serotonin |
5-HT2A / HTR2A |
NM_003950 |
| CHO-K1/5-HT2B |
Serotonin |
5-HT2B / HTR2B |
NM_000867 |
| 293/5-HT2B |
Serotonin |
5-HT2B / HTR2B |
NM_000867 |
| CHO-K1/5-HT2C |
Serotonin |
5-HT2C / HTR2C |
NM_000868 |
| 293/5-HT2C |
Serotonin |
5-HT2C / HTR2C |
NM_000868 |
| CHO-K1/SST2/Gα15 |
Somatostatin |
SST2 |
NM_001050 |
| CHO-K1/SST3/Gα15 |
Somatostatin |
SST3 |
NM_001051 |
| CHO-K1/SST4/Gα15 |
Somatostatin |
SST4 |
NM_001052 |
| CHO-K1/SST5/Gα15 |
Somatostatin |
SST5 |
NM_001053 |
| CHO-K1/PRLHR |
Prolactin Releasing Peptide |
PRLHR |
NM_004248 |
| 1321N1/P2Y2 |
Purinergic |
P2Y2 |
NM_176071 |
| 1321N1/P2Y4 |
Purinergic |
P2Y4 |
NM_002565 |
| 1321N1/P2Y11 |
Purinergic |
P2Y11 |
NM_002566 |
| 1321N1/P2Y12/Gα15 |
Purinergic |
P2Y12 |
NM_176876 |
| CHO-K1/NK1 |
Tachykinin |
NK1 / TACR1 |
NM_001058 |
| CHO-K1/NK2 |
Tachykinin |
NK2 / TACR2 |
NM_001057 |
| CHO-K1/NK3 |
Tachykinin |
NK3 / TACR3 |
NM_001059 |
| CHO-K1/TRH1 |
Thyrtropin-releasing Hormone |
TRH1 |
NM_003301 |
| CHO-K1/UTR2/Gα15 |
Urotensin |
UTR2 |
NM_018949 |
| CHO-K1/V1A |
Vasopressin |
V1A / AVPR1A |
NM_000706 |
| CHO-K1/V1B |
Vasopressin |
V1B / AVPR1B |
NM_000706 |
| CHO-K1/V2/Gα15 |
Vasopressin |
V2 / AVPR2 |
NM_000054 |
| CHO-K1/PAC1/Gα15 |
VIP/PACAP |
PAC1 |
NM_001118 |
| CHO-K1/VPAC1/Gα15 |
VIP/PACAP |
VPAC1 |
NM_004624 |
| CHO-K1/VPAC2/Gα15 |
VIP/PACAP |
VPAC2 |
NM_003382 |
All the GPCRs are available as Ready-to-UseTM frozen cells.
A part of the GPCRs are available as Membrane Preparations.
Ion Channels
Name |
Type |
Channel |
Accession Number |
| CHO-K1/hERG |
Potassium, voltage-gated |
hERG (Kv11.1) |
NM_000238.2 |
| HEK293/hERG |
Potassium, voltage-gated |
hERG (Kv11.1) |
NM_000238.2 |
| HEK293/Kv1.5 |
Potassium, voltage-gated |
Kv1.5 |
NM_002234 |
Custom Stable Cell Line Services:
| Cat. No. |
Service |
Price (USD) |
SC1394 |
Custom Stable Cell Line Service |
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Related Services:
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Email: bioassay@genscript.com |
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Phone: 1-877-436-7274 (Toll-Free), 1-732-885-9188 |
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Fax: 1-732-210-0262, 1-732-885-5878 |
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