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GPCR & Ion Channel Stable Cell Line Collection

GenScript offers a wide selection of GPCR and ion channel stable cell lines exclusively for assay services. In addition, GenScript offers one-stop assay reagent preparations for your compound screening/profiling: Ready-to-UseTM Frozen Cells, Membrane Preparations, and Custom Stable Cell Line Service.

GPCRs

Name
GPCR Family
Receptor
Accession Number
CHO-K1/M1 Acetylcholine (muscarinic) M1 / CHRM1
NM_000738
CHO-K1/M3 Acetylcholine (muscarinic) M3 / CHRM3
NM_000740
CHO-K1/M5 Acetylcholine (muscarinic) M5 / CHRM5
NM_012125
CHO-K1/ADORA1/Gα15 Adenosine ADORA1
NM_000674
CHO-K1/ADORA2B/Gα15 Adenosine ADORA2B
NM_000675
CHO-K1/ADRA1A Adrenoceptors ADRA1A
NM_000680
CHO-K1/ADRA1B Adrenoceptors ADRA1B
NM_000679
CHO-K1/ADRA1D Adrenoceptors ADRA1D
NM_000678
CHO-K1/ADRA2A/Gα15 Adrenoceptors ADRA2A
NM_000681
CHO-K1/ADRB1/Gα15 Adrenoceptors ADRB1
NM_000684
CHO-K1/ADRB2/Gα15 Adrenoceptors ADRB2
NM_000024
293/ADRB3/CRE-Luc Adrenoceptors ADRB3
NM_000025
CHO-K1/C5a/Gα15 Anaphylotoxin C5a / C5AR1
NM_001736
CHO-K1/BB2 Bombesin BB2
NM_005314
CHO-K1/BB3 Bombesin BB3
NM_001727
CHO-K1/B2/Gα15 Bradykinin B2
NM_000623
CHO-K1/CALCR/Gα15 Calcitonin CALCR
NM_001742.2
CHO-K1/CNR1/Gα15 Cannabinoid CNR1 / CB1
NM_016083
CHO-K1/CMKLR1/Gα15 Chemoattractant CMKLR1
NM_004072
CHO-K1/CCKA/Gα15 Cholecystokinin CCKA
NM_000730
CHO-K1/CCKB Cholecystokinin CCKB
NM_176875
CHO-K1/CRF1/Gα15 Corticotropin Releasing Factor CRF1
NM_004382
CHO-K1/CRF2/Gα15 Corticotropin Releasing Factor CRF2
NM_001883
CHO-K1/D2/Gα15 Dopamine D2
NM_000795
CHO-K1/D2s/Gα15 Dopamine D2S
NM_016574
CHO-K1/D5/Gα15 Dopamine D5
NM_000798
CHO-K1/EDNRA Endothelin EDNRA
NM_000795
CHO-K1/EDNRB Endothelin EDNRB
NM_000115
CHO-K1/GPR40-GFP Free Fatty Acid FFA1 / GPR40
NM_005303
CHO-K1/GPR40/Gα15 Free Fatty Acid FFA1 / GPR40
NM_005303
CHO-K1/GAL1/Gα15 Galanin GAL1
NM_001480
CHO-K1/GAL2 Galanin GAL2
NM_003857
CHO-K1/GHSR Ghrelin GHSR
NM_198407
293/GHRH/Gα15 Glucagon GHRH
NM_000823
CHO-K1/GLP2/Gα15 Glucagon GLP2
NM_004246
CHO-K1/SCTR/Gα15 Glucagon SCTR
NM_002980
293/H1 Histamine H1
NM_000861
CHO-K1/H2/Gα15 Histamine H2
NM_022304
CHO-K1/H3/Gα15 Histamine H3
NM_007232
CHO-K1/H4/Gα15 Histamine H4
NM_021624
CHO-K1/KISS1 KiSS1-derived peptide KiSS1 / GPR54
NM_032551
293/MCH1 Melanin-concentrating Hormone MCH1
NM_005297
CHO-K1/MCH2 Melanin-concentrating Hormone MCH2
NM_032503
CHO-K1/MC2/Gα15 Melanocortin MC2
NM_000529
CHO-K1/MC3/Gα15 Melanocortin MC3
NM_019888
293/MC3/CRE-Luc Melanocortin MC3
NM_019888
CHO-K1/MC4/Gα15 Melanocortin MC4
NM_005912
CHO-K1/MT2/Gα15 Melatonin MT2
NM_005959
CHO-K1/NMU1 Neuromedin U NMU1
NM_006056
CHO-K1/GPR103/Gα15 Neuropeptide GPR103
NM_198179
CHO-K1/NPS1a/Gα15 Neuropeptide S NPS1a
NM_207172
CHO-K1/NTS1 Neurotensin NTS1
NM_002531
CHO-K1/FPRL1/Gα15 N-Formyl Peptide FPRL1
NM_001462
CHO-K1/OPRD1/Gα15 Opioid OPRD1
NM_000911
CHO-K1/OPRK1/Gα15 Opioid OPRK1
NM_000912
CHO-K1/OPRM1/Gα15 Opioid OPRM1
NM_000914
CHO-K1/OX1 Orexin OX1
NM_001525
CHO-K1/OX2 Orexin OX2
NM_001526
CHO-K1/OXTR Oxytocin OT / OXTR
NM_000916
CHO-K1/PTH1/Gα15 Parathyroid Hormone PTH1
NM_000316
293/PTH2/CRE-Luc Parathyroid Hormone PTH2
NM_005048
CHO-K1/PTAFR Platelet Activating Factor PAF / PTAFR
NM_000952
293/FP/Gα15 Prostanoid FP / PTGFR
NM_000952
293/PTGER1 Prostanoid EP1 / PTGER1
NM_000955.2
CHO-K1/PTGER2/Gα15 Prostanoid EP2 / PTGER2
NM_000956
CHO-K1/IP1/Gα15 Prostanoid IP1 / PTGIR
NM_000960
293/TP Prostanoid TP / TBXA2R
NM_001060
CHO-K1/PAR4 Proteinase-activated Receptor PAR4 / F2RL3
NM_003950
CHO-K1/5-HT1A/Gα15 Serotonin 5-HT1A / HTR1A
NM_000524
CHO-K1/5-HT1D/Gα15 Serotonin 5-HT1D / HTR1D
NM_000864
CHO-K1/5-HT2A Serotonin 5-HT2A / HTR2A
NM_003950
CHO-K1/5-HT2B Serotonin 5-HT2B / HTR2B
NM_000867
293/5-HT2B Serotonin 5-HT2B / HTR2B
NM_000867
CHO-K1/5-HT2C Serotonin 5-HT2C / HTR2C
NM_000868
293/5-HT2C Serotonin 5-HT2C / HTR2C
NM_000868
CHO-K1/SST2/Gα15 Somatostatin SST2
NM_001050
CHO-K1/SST3/Gα15 Somatostatin SST3
NM_001051
CHO-K1/SST4/Gα15 Somatostatin SST4
NM_001052
CHO-K1/SST5/Gα15 Somatostatin SST5
NM_001053
CHO-K1/PRLHR Prolactin Releasing Peptide PRLHR
NM_004248
1321N1/P2Y2 Purinergic P2Y2
NM_176071
1321N1/P2Y4 Purinergic P2Y4
NM_002565
1321N1/P2Y11 Purinergic P2Y11
NM_002566
1321N1/P2Y12/Gα15 Purinergic P2Y12
NM_176876
CHO-K1/NK1 Tachykinin NK1 / TACR1
NM_001058
CHO-K1/NK2 Tachykinin NK2 / TACR2
NM_001057
CHO-K1/NK3 Tachykinin NK3 / TACR3
NM_001059
CHO-K1/TRH1 Thyrtropin-releasing Hormone TRH1
NM_003301
CHO-K1/UTR2/Gα15 Urotensin UTR2
NM_018949
CHO-K1/V1A Vasopressin V1A / AVPR1A
NM_000706
CHO-K1/V1B Vasopressin V1B / AVPR1B
NM_000706
CHO-K1/V2/Gα15 Vasopressin V2 / AVPR2
NM_000054
CHO-K1/PAC1/Gα15 VIP/PACAP PAC1
NM_001118
CHO-K1/VPAC1/Gα15 VIP/PACAP VPAC1
NM_004624
CHO-K1/VPAC2/Gα15 VIP/PACAP VPAC2
NM_003382

All the GPCRs are available as Ready-to-UseTM frozen cells.
A part of the GPCRs are available as Membrane Preparations.

Ion Channels

Name
Type
Channel
Accession Number
CHO-K1/hERG Potassium, voltage-gated hERG (Kv11.1)
NM_000238.2
HEK293/hERG Potassium, voltage-gated hERG (Kv11.1)
NM_000238.2
HEK293/Kv1.5 Potassium, voltage-gated Kv1.5
NM_002234

Custom Stable Cell Line Services:

Cat. No. Service
Price (USD)
SC1394
Custom Stable Cell Line Service

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