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GPCR and Ion Channel Stable Cell Lines

GenScript offers a wide selection of GPCR and ion channel stable cell lines. Proprietary codon optimization and vector design technologies enable GenScript to overcome low functional expression of protein at the cell surface. All of the cell lines have been optimized for S/B ratio in calcium flux assay or other assays and shown stability after over 16 passages.

Tailored to your specifications, GenScript Custom Stable Cell Line Service is available.

Key Features:

  • High functional expression of proteins at the cell surface
  • Stable cell lines for increased reliability and reproducibility
  • All ion channel stable cell lines are validated by manual patch clamp, and Qpatch
  • Flexible functional readouts are available

GPCR Stable Cell Lines:

Cat. No. Name Family Receptor
Size   
Price (USD)
Selected
CHO-K1/M1 Acetylcholine (muscarinic) M1
2 vials
$11600.00
HEK293/M1 Acetylcholine (muscarinic) M1
2 vials
CHO-K1/M3 Acetylcholine (muscarinic) M3
2 vials
$11600.00
CHO-K1/M5 Acetylcholine (muscarinic) M5
2 vials
$11600.00
CHO-K1/A1/Gα15 Adenosine A1
2 vials
$11600.00
CHO-K1/ADRA1A Adrenoceptors ADRA1A
2 vials
$11600.00
CHO-K1/ADRA1B Adrenoceptors ADRA1B
2 vials
$11600.00
CHO-K1/ADRB1/Ga15 Adrenoceptors ADRB1
2 vials
$11600.00
CHO-K1/ADRB2/Gα15 Adrenoceptors ADRB2
2 vials
$11600.00
CHO-K1/BB2 Bombesin BB2
2 vials
$11600.00
CHO-K1/BB3 Bombesin BB3
2 vials
$11600.00
CHO-K1/B2/Gα15 Bradykinin B2
2 vials
$11600.00
CHO-K1/CALCR/Gα15 Calcitonin CALCR
2 vials
$11600.00
CHO-K1/CMKLR1/Gα15 Chemoattractant CMKLR1
2 vials
$11600.00
CHO-K1/CCKA/Gα15 Cholecystokinin CCKA
2 vials
$11600.00
CHO-K1/CCKB Cholecystokinin CCKB
2 vials
$11600.00
CHO-K1/CRF2/Gα15 Corticotropin Releasing Factor CRF2
2 vials
$11600.00
HEK293/D1/CRE/β-Lac Dopamine D1
2 vials
CHO-K1/D2/Gα15 Dopamine D2
2 vials
$11600.00
HEK293/D2/Gα15 Dopamine D2
2 vials
CHO-K1/D2s/Gα15 Dopamine D2s
2 vials
$11600.00
HEK293/D5/CRE/β-Lac Dopamine D5
2 vials
CHO-K1/EDNRA Endothelin EDNRA
2 vials
$11600.00
CHO-K1/EDNRB Endothelin EDNRB
2 vials
$11600.00
CHO-K1/GPR40-GFP Free Fatty Acid FFA1/GPR40
2 vials
$11600.00
CHO-K1/GPR40/Gα15 Free Fatty Acid FFA1/GPR40
2 vials
$11600.00
HEK293/GPR40/NFAT/β-Lac Free Fatty Acid FFA1/GPR40
2 vials
CHO-K1/GAL1/Gα15 Galanin GAL1
2 vials
$11600.00
CHO-K1/GAL2 Galanin GAL2
2 vials
$11600.00
CHO-K1/GHSR Ghrelin GHSR
2 vials
$11600.00
CHO-K1/GLP2/Gα15 Glucagon GLP2
2 vials
$11600.00
HEK293/GnRHR/NFAT/β-Lac Gonadotropin-Releasing Hormone GnRH
2 vials
293/H1 Histamine H1
2 vials
$11600.00
CHO-K1/H2/Gα15 Histamine H2
2 vials
$11600.00
HEK293/H2/CRE/Luc Histamine H2
2 vials
HEK293/H3/Gα15 Histamine H3
2 vials
HEK293/H4/Gα16 Histamine H4
2 vials
CHO-K1/H4/Gα15 Histamine H4
2 vials
$11600.00
293/MCH1 Melanin-concentrating Hormone MCH1
2 vials
$11600.00
HEK293/MCH2 Melanin-concentrating Hormone MCH2
2 vials
CHO-K1/MCH2 Melanin-concentrating Hormone MCH2
2 vials
$11600.00
CHO-K1/MC4/Gα15 Melanocortin MC4
2 vials
$11600.00
CHO-K1/MT2/Gα15 Melatonin MT2
2 vials
$11600.00
CHO-K1/NMU1 Neuromedin U NMU1
2 vials
$11600.00
CHO-K1/GPR103/Gα15 Neuropeptide GPR103
2 vials
$11600.00
CHO-K1/NTS1 Neurotensin NTS1
2 vials
$11600.00
CHO-K1/FPRL1/Gα15 N-Formyl Peptide FPRL1
2 vials
$11600.00
CHO-K1/OPRK1/Gα15 Opioid OPRK1
2 vials
$11600.00
CHO-K1/OPRM1/Gα15 Opioid OPRM1
2 vials
$11600.00
CHO-K1/OX1 Orexin OX1
2 vials
$11600.00
CHO-K1/OX2 Orexin OX2
2 vials
$11600.00
CHO-K1/OXTR Oxytocin OT/OXTR
2 vials
$11600.00
CHO-K1/PTH1/Gα15 Parathyroid Hormone PTH1
2 vials
$11600.00
HEK293/PTHR1/CRE/β-Lac Parathyroid Hormone PTH1
2 vials
HEK293/PTHR2/CRE/β-Lac Parathyroid Hormone PTH2
2 vials
CHO-K1/PTAFR Platelet Activating Factor PTAFR
2 vials
$11600.00
HEK293/PAFR/NFAT/β-Lac Platelet Activating Factor PTAFR
2 vials
293/FP/Gα15 Prostanoid FR
2 vials
$11600.00
CHO-K1/IP1/Gα15 Prostanoid IP1
2 vials
$11600.00
293/PTGER1 Prostanoid PTGER1
2 vials
$11600.00
CHO-K1/PTGER2/Gα15 Prostanoid PTGER2
2 vials
$11600.00
293/TP Prostanoid TP
2 vials
$11600.00
CHO-K1/PAR4 Proteinase-activated Receptor PAR4
2 vials
$11600.00
CHO-K1/5-HT2A Serotonin 5-HT2A
2 vials
$11600.00
CHO-K1/5-HT2B Serotonin 5-HT2B
2 vials
$11600.00
CHO-K1/5-HT2C Serotonin 5-HT2C
2 vials
$11600.00
CHO-K1/SST3/Gα15 Somatostatin SST3
2 vials
$11600.00
CHO-K1/SST5/Gα15 Somatostatin SST5
2 vials
$11600.00
1321N1/P2Y2 Purinergic P2Y2
2 vials
$11600.00
1321N1/P2Y4 Purinergic P2Y4
2 vials
$11600.00
1321N1/P2Y11 Purinergic P2Y11
2 vials
$11600.00
HEK293/SPR Tachykinin NK1/SPR
2 vials
CHO-K1/NK1 Tachykinin NK1/SPR
2 vials
$11600.00
CHO-K1/NK2 Tachykinin NK2
2 vials
$11600.00
CHO-K1/NK3 Tachykinin NK3
2 vials
$11600.00
CHO-K1/TRH1 Thyrtropin-releasing Hormone TRH1
2 vials
$11600.00
CHO-K1/V1A Vasopressin V1A
2 vials
$11600.00
CHO-K1/V1B Vasopressin V1B
2 vials
$11600.00
CHO-K1/V2/Gα15 Vasopressin V2
2 vials
$11600.00
CHO-K1/CRE/Luc Host Cell Line N/A
2 vials
$11600.00
293/CRE/Luc Host Cell Line N/A
2 vials
$11600.00
* The stable cell lines can be treated to produce Ready-to-UseTM frozen cells.

Custom Stable Cell Line Services:

Cat. No. Service
Price (USD)
SC1394
Custom Stable Cell Line Service

Email: bioassay@genscript.com
Phone: 1-877-436-7274 (Toll-Free), 1-732-885-9188
Fax: 1-732-210-0262, 1-732-885-5878