Dermorphin Analog

*This product has been discontinued!*

The dermorphin-derived peptide [Dmt1] dermorphin analog labels m-opioid receptors with high affinity and selectivity in receptor binding assays. In mice, radiant heat tail-flick assays, [Dmt1] dermorphin analog produces profound spinal and supraspinal analgesia, being approximately 5000 and 100 times more potent respectively than morphine in causing these analgesia on a molar basis. When administered systemically, [Dmt1] dermorphin analog has been shown to be over 200 times more potent than morphine.

Cat. No.	RP13522
Size	Buy in bulk

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Overview Properties

Description

The dermorphin-derived peptide [Dmt1] dermorphin analog labels m-opioid receptors with high affinity and selectivity in receptor binding assays. In mice, radiant heat tail-flick assays, [Dmt1] dermorphin analog produces profound spinal and supraspinal analgesia, being approximately 5000 and 100 times more potent respectively than morphine in causing these analgesia on a molar basis. When administered systemically, [Dmt1] dermorphin analog has been shown to be over 200 times more potent than morphine.

Overview

Sequence	TYR-d-ARG-PHE-SAR-TYR-PRO-SER-NH₂
Molecular Formula	C₄₄H₅₉N₁₁O₁₀
C Terminal	NH₂
Molecular Weight	901.43

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Properties

Purity	> 95%
Solubility	Dermorphin analog is soluble in water. The contents of this vial have been accurately determined. Both the stopper and the vial have been siliconized. Do not attempt to weigh out a smaller portion of the contents.
Storage	Before use, store dermorphin analog in the DRY form at 0-5°C. For best and most repeatable results, rehydrate the peptide immediately before use. Do not re-freeze any unused portions.

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